Aprepitant:anti-P
補充止吐
⑴ Motion sickness, Meniere’s disease: H1 & M3 antagonist
⑵ 化療: NK1 Receptor antagonist, 5-HT3 antagonist, Corticosteroids, cannabinoids, Anti-substance P
⑶ 手術: 5-HT3 & Dopamine antagonist, corticosteroids
⑷ 孕吐: Doxylamine + pyridoxine
NK1受體抑制劑機轉:阻止大腦中樞的substance P作用在NK-1受體。藥:Aprepitant、netupitant、rolapitant(三個都是口服)。
26.用於預防化療(chemotherapy)引起之噁心及嘔吐之藥物Aprepi..-阿摩線上測驗