55. 下圖losartan結構中之取代基分別為: (A)R1=t..-阿摩線上測驗
10F YUI_1222 高三下 (2018/12/22)
Phenyl ortho-carboxylate - Temisartan Phenyl ortho-tetrazole - Losartan,Valsartan(沒有imidazole),Irbsartan,Candesartan 對AT1受體選擇性 candesartan>irbesartan>telmisartan=valsartan=Exp3174>losartan 比較 對cox2 抑制選擇性 Etoricoxib>rofecoxib>valdecoxib>celecoxib 雜環 bipyridine furanone isoxazole pyrazole lactone |
11F
|
12F
|