73.有關藥物基因檢測結果與藥品及其效果或不良反應的配對,下列何者正確?
(A)CYP2C19 rapid metabolizer:clopidogrel-antiplatelet activity 不佳
(B)CYP2D6 slow metabolizer:codeine-analgesic effect 較佳
(C)HLA-B*1502:allopurinol-Stevens-Johnson Syndrome 機率增加
(D)thiopurine methyltransferase(TPMT)slow metabolizer:azathioprine-pancytopenia 機率增加
答案:登入後查看
統計: A(3), B(0), C(6), D(18), E(0) #3972582
統計: A(3), B(0), C(6), D(18), E(0) #3972582
詳解 (共 5 筆)
#7525200
(A)Clopidogrel為Prodrug,透過CYP2C19轉化為活性態,若為CYP2C19 rapid metabolizer則抗血小板能力會更好
(B)Codeine為Prodrug,透過CYP2D6轉化為活性態,若為CYP2D6 slow metabolizer則鎮痛效果較差
(C)Allopurinol是HLA-B*5801
0
0