72.下列何組藥品交互作用的機制,不屬於藥動學交互作用?
(A)theophylline-amiodarone
(B)alcohol-disulfiram
(C)allopurinol-mercaptopurine
(D)digoxin-hydrochlorothiazide
答案:登入後查看
統計: A(333), B(1256), C(526), D(1909), E(0) #2404278
統計: A(333), B(1256), C(526), D(1909), E(0) #2404278
詳解 (共 10 筆)
#4493805
藥動學: 與ADME有關 (吸收分布代謝排除)
藥效學: 藥理作用
digoxin-hydrochlorothiazide: TZD副作用低血鉀導致digoxin (Na+/K+-ATPase)毒性上升
31
6
#5512691
酒癮
|
乙醇Ethanol |
→ADH醇脫氫酶→
|
乙醛acetaldehyde(嘔吐頭痛) |
→ALDH醛脫氫酶→
|
醋酸Acetate |
|
甲醇Methanol |
甲醛formaldehyde |
甲酸Formate(毒) |
||
|
|
X↑Fomepizole (解酒扶ME) |
|
X↑disulfram:酒癮治療, 使乙醛滯留,人不舒服而停止喝酒 |
|
ADH alcohol dehydroganase乙醇脫氫酶
ALDH aldehyde dehydroganase醛脫氫酶
甲醇中毒:用乙醇IV解毒,乙醇AOH親和力較好使先代謝
乙醇:blockouts抑制NMDA受體
13
0