15 下述那一個副交感神經作用藥物,其對Nicotinic receptor 之作用最強?
(A) Pilocarpine
(B) Carbachol
(C) Bethanechol
(D) Methacholine
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統計: A(46), B(189), C(50), D(91), E(0) #443760
統計: A(46), B(189), C(50), D(91), E(0) #443760
詳解 (共 3 筆)
#1305341
(A) Pilocarpine 蕈毒鹼(M)
(B) Carbachol 無選擇性(M、N)
(C) Bethanechol 蕈毒鹼(M)
(D) Methacholine 蕈毒鹼(M)
(B) Carbachol 無選擇性(M、N)
(C) Bethanechol 蕈毒鹼(M)
(D) Methacholine 蕈毒鹼(M)
9
0
#1237499
27 下列擬副交感神經作用劑中,何者不會被膽鹼酯酶(cholinesterase)水解,對於尼古丁(nicotinic)及蕈毒鹼受體(muscarinic receptor)皆有作用?
(A) acetylcholine
(B) methacholine
(C) carbachol
(D) bethanechol
答案C
6
0
#802087
A cholinergic (parasympathomimetic) agent. Carbachol acts directly to stimulate muscarinic (smooth muscle) and nicotinic (autonomic ganglia) receptors and indirectly to inhibit cholinesterase enzyme activity. Carbachol is resistant to hydrolysis by cholinesterases.
2
0