74 下列何種藥物不需經過bioactivation 即有抗癌活性?
(A) 6-Mercaptopurine
(B) 5-FU
(C) Doxorubicin
(D) Cyclophosphamide
答案:登入後查看
統計: A(99), B(145), C(740), D(174), E(0) #416508
統計: A(99), B(145), C(740), D(174), E(0) #416508
詳解 (共 4 筆)
#1025626
Azathioprine (AZA) ---> 6-MP ---> 6-TNG + 6-MMPR + 6-thio-ITP
Capecitabine ---> 5-FU ---> FdUMP (fluorodeoxyuridine monophosphate)
Cyclophosphamide ---> 4-Hydroxycyclophosphamide
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0
#1025627
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#843252
Cyclophosphamide oral and injection 一種prodrug 且可口服 在體內經肝臟 P-450代謝後形成4-hydroxycyclophosphamide...
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