74 下列何種藥物不需經過bioactivation 即有抗癌活性?
(A) 6-Mercaptopurine
(B) 5-FU
(C) Doxorubicin
(D) Cyclophosphamide

答案:登入後查看
統計: A(99), B(145), C(740), D(174), E(0) #416508

詳解 (共 4 筆)

#1025626
Azathioprine (AZA) ---> 6-MP ---> 6-TNG + 6-MMPR + 6-thio-ITP 
Capecitabine  ---> 5-FU  ---> FdUMP (fluorodeoxyuridine monophosphate)
Cyclophosphamide --->  4-Hydroxycyclophosphamide
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#1025627
%25252254c681aa87a22.jpg%252522.png
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#843252
Cyclophosphamide oral and injection 一種prodrug 且可口服 在體內經肝臟 P-450代謝後形成4-hydroxycyclophosphamide...
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#6533542
抗癌 —---------------...




































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