34.下述那一個化合物對於中樞神經GABA-A受體最具有選擇性拮抗作用?
(A)d-Tubocurarine
(B)Bicuculline
(C)Prazosin
(D)Ketanserin
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統計: A(386), B(2069), C(126), D(562), E(0) #415076
統計: A(386), B(2069), C(126), D(562), E(0) #415076
詳解 (共 6 筆)
#895314
GABAa receptor allosteric moclulator:(異位作用)
負向:picrotoxin.phenyleneterazole----CNS興奮
正向:BZD.Barbiturates------CNS抑制
GABAa recptor:(直接作用)
作用劑:Muscimol
拮抗劑:Bicuclline
144
2
#799213
Bicuculline is a light-sensitive competitive antagonist of GABAA receptors.
11
1